Azasetron hydrochloride ( Azasetron hydrochloride;Y 25130; Y-25130; Y25130. )

产品货号. M10908 CAS No. 123040-16-4

COA

Datasheet

HNMR

HPLC

MSDS

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产品名称

Azasetron hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Azasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.
产品描述

Azasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.Azasetron inhibited the specific binding of [3H]quipazine to 5-HT3 receptors at the synaptic membranes of the rat cerebral cortex.
同义词

Azasetron hydrochloride;Y 25130; Y-25130; Y25130.
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT3
研究领域

Neurological Disease
适应症

——

CAS Number

123040-16-4
分子量

386.27
分子式

C17H20ClN3O3·HCl
纯度

>98%(HPLC)
溶解度

Water: 3 mg/mL (7.76 mM)
SMILES

c1(cc(C(N[C@@H]2CN3CCC2CC3)=O)c2c(c1)N(C)C(=O)CO2)Cl.Cl
化学全称

2H-1,4-Benzoxazine-8-carboxamide, 3,4-dihydro-N-1-azabicyclo(2.2.2)oct-3-yl-6-chloro-4-methyl-3-oxo-, monohydrochloride

1.Katayama K, et al. Jpn J Pharmacol. 1997 Apr;73(4):357-60.

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产品手册

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